SCHEMBL8515898

SCHEMBL8515898

Cc1c(-c2ccc(Cc3ccc(OC(F)(F)F)cc3)cc2)nc2cc(Cl)ccc2c1OP(=O)(O)O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
DHODH Q02127 3/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.38
TRPM8 Q7Z2W7 1/20 0.37
P2RY14 Q15391 1/20 0.37
PTGFR P43088 2/20 0.35
SCN10A Q9Y5Y9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515893 0.93 CYP3A4 (0.44) CYP3A4DHODHPTGDR2TRPM8P2RY14
SCHEMBL8514061 0.84 DHODH (0.42) CYP3A4DHODHPTGDR2TRPM8P2RY14
SCHEMBL8514758 0.80 DHODH (0.44) DHODHPTGFRSCN10A
SCHEMBL8515434 0.79 HSD17B10 (0.43) CYP3A4DHODH
SCHEMBL8514251 0.73 PDE10A (0.44) DHODHTRPM8PTGFR
SCHEMBL8514255 0.73 PDE10A (0.44) DHODHTRPM8PTGFR
SCHEMBL8515384 0.72 ACP1 (0.44) DHODHPTGFRSCN10A
SCHEMBL8512120 0.70 SCN9A (0.45) DHODHTRPM8PTGFR
SCHEMBL8534985 0.67 MAPK8 (0.40) CYP3A4DHODHPTGDR2
SCHEMBL8535303 0.66 MAT2A (0.55) CYP3A4PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed