SCHEMBL8517876

SCHEMBL8517876

C=CCc1ccc(-c2ccc(C#CC(C)O)cn2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.35
SMN1; SMN2 Q16637 7/20 0.35
NPC1 O15118 7/20 0.35
MAPT P10636 3/20 0.35
STAT3 P40763 1/20 0.35
ATM Q13315 1/20 0.35
TP53 P04637 1/20 0.35
KDM4E B2RXH2 5/20 0.34
ALDH1A1 P00352 5/20 0.34
HPGD P15428 5/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
GRM5 P41594 3/20 0.34
MITF O75030 1/20 0.34
KLF5 Q13887 1/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
MAPK1 P28482 1/20 0.34
CYP11B1 P15538 1/20 0.34
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517335 0.84 CYP2D6 (0.44) RAB9ANPC1MAPTTP53KDM4E
SCHEMBL8517798 0.84 ALDH1A1 (0.39) SMN1; SMN2MAPTTP53KDM4EALDH1A1
SCHEMBL8517840 0.82 ACACB (0.41) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL9288296 0.80 GRM5 (0.32) RAB9AMAPTKDM4EALDH1A1HPGD
SCHEMBL8517733 0.79 ACACB (0.40) SMN1; SMN2MAPTTP53KDM4EALDH1A1
SCHEMBL4890255 0.77 L3MBTL1 (0.50) RAB9ASMN1; SMN2NPC1MAPTKDM4E
SCHEMBL8518327 0.77 ACACB (0.40) RAB9ASMN1; SMN2NPC1MAPTTP53
SCHEMBL7557671 0.77 RAB9A (0.33) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL7552712 0.76 L3MBTL1 (0.33) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL9288293 0.76 GRM5 (0.33) RAB9ASMN1; SMN2NPC1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed