SCHEMBL8517823

SCHEMBL8517823

C[Si](C)(COc1ccc(O)cc1)c1ccc(N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.44
TSHR P16473 1/20 0.44
THRB P10828 2/20 0.43
HIF1A Q16665 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CA3 P07451 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
CA6 P23280 1/20 0.43
CASP1 P29466 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CA14 Q9ULX7 1/20 0.43
ESR1 P03372 1/20 0.43
CYP19A1 P11511 1/20 0.43
ESR2 Q92731 1/20 0.43
GAA P10253 3/20 0.42
LTA4H P09960 3/20 0.41
APP P05067 2/20 0.40
MAOB P27338 4/20 0.40
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8374301 0.85 ESR2 (0.50) ALDH1A1ESR1ESR2GAALTA4H
SCHEMBL8887466 0.83 CYP1A2 (0.42) ALDH1A1HSD17B10LTA4HAPPMAOB
SCHEMBL8444609 0.83 LMNA (0.52) HIF1AESR1CYP19A1ESR2GAA
SCHEMBL7520674 0.77 NR1H4 (0.52) ALDH1A1ALOX15HSD17B10GAAMAPT
SCHEMBL8443089 0.74 LTA4H (0.52) HIF1AESR1ESR2LTA4HAPP
SCHEMBL12660720 0.74 TDP1 (0.58) TDP1TSHRALDH1A1CYP3A4HSD17B10
SCHEMBL6054922 0.72 CA2 (0.45) TDP1TSHRHIF1AALDH1A1CYP3A4
SCHEMBL8518289 0.71 ESR2 (0.50) ALDH1A1ESR1ESR2GAALTA4H
SCHEMBL2194744 0.71 TDP1 (0.54) TDP1TSHRALDH1A1CYP3A4HSD17B10
SCHEMBL7517793 0.70 TSHR (0.34) TSHRCASP1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-03-10 EP disclosed
WO-1997041129-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-11-06 WO disclosed