SCHEMBL8524211

SCHEMBL8524211

CC1CC2N(C)C(=O)CC(Cc3ccccc3)[C@]2(C)[C@@H]2CC[C@]3(C)CCC[C@H]3[C@H]12

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 7/20 0.34
SRD5A2 P31213 5/20 0.34
CYP19A1 P11511 8/20 0.32
OPRK1 P41145 2/20 0.32
CHRM5 P08912 1/20 0.32
CHRM3 P20309 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523844 0.86 CYP19A1 (0.33) SRD5A1SRD5A2CYP19A1
SCHEMBL8637459 0.83 ALDH1A1 (0.35) SRD5A1SRD5A2
SCHEMBL8633124 0.82 SRD5A1 (0.33) SRD5A1SRD5A2CYP19A1
SCHEMBL8523847 0.80 SRD5A1 (0.36) SRD5A1SRD5A2CYP19A1
SCHEMBL8523105 0.79 SHBG (0.36) SRD5A1SRD5A2
SCHEMBL8522986 0.78 SRD5A1 (0.35) SRD5A1SRD5A2
SCHEMBL8523422 0.77 MBOAT4 (0.34) SRD5A1SRD5A2
SCHEMBL8639064 0.77 SRD5A1 (0.34) SRD5A1SRD5A2
SCHEMBL8642307 0.75 SRD5A1 (0.32) SRD5A1SRD5A2
SCHEMBL8996754 0.75 SRD5A1 (0.31) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP claimed
WO-1998009632-A1 METHODS AND COMPOSITIONS FOR TREATING PRETERM LABOR MERCK & CO., INC. (US) 1998-03-12 WO claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1998009632-A1 METHODS AND COMPOSITIONS FOR TREATING PRETERM LABOR MERCK & CO., INC. (US) 1998-03-12 WO disclosed