SCHEMBL8524419

SCHEMBL8524419

CC1(C)CCC(=O)Nc2ccc(C(=O)CCl)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
MAPT P10636 1/20 0.49
HDAC3 O15379 5/20 0.43
HDAC4 P56524 5/20 0.43
HDAC1 Q13547 5/20 0.43
HDAC2 Q92769 5/20 0.43
HDAC8 Q9BY41 5/20 0.43
HDAC6 Q9UBN7 5/20 0.43
HDAC9 Q9UKV0 5/20 0.43
MET P08581 4/20 0.39
CYP3A4 P08684 2/20 0.39
INSR P06213 2/20 0.39
CYP26A1 O43174 1/20 0.39
CYP26B1 Q9NR63 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
USP2 O75604 1/20 0.38
F2 P00734 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6450714 0.86 HDAC3 (0.56) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL8524882 0.82 ALDH1A1 (0.47) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL8525367 0.81 SMN1; SMN2 (0.38) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL9184645 0.77 CYP3A4 (0.59) ALDH1A1CYP3A4CYP26A1CYP26B1RARA
SCHEMBL6218261 0.76 HDAC6 (0.54) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL8524985 0.76 ALDH1A1 (0.43) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL1145012 0.76 ALDH1A1 (0.55) ALDH1A1MAPTHDAC3HDAC4HDAC1
SCHEMBL5680486 0.76 PGR (0.50) ALDH1A1MAPTSMN1; SMN2USP2F2
SCHEMBL15304426 0.74 CYP3A4 (0.50) ALDH1A1MAPTMETCYP3A4INSR
SCHEMBL11470235 0.74 HDAC6 (0.54) ALDH1A1MAPTHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed