SCHEMBL8524922

SCHEMBL8524922

COc1ccc(-n2c(C)ccc2NS(=O)(=O)c2ccccc2)cc1Cl.COc1ccc(-n2c(C)ccc2NS(=O)(=O)c2ccccc2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
MAPT P10636 4/20 0.46
LMNA P02545 3/20 0.46
HTT P42858 2/20 0.46
THRB P10828 1/20 0.46
HPGD P15428 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
TSHR P16473 3/20 0.42
POLB P06746 3/20 0.42
HSD17B10 Q99714 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PTGS1 P23219 2/20 0.40
PTGS2 P35354 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8505452 0.94 HPGD (0.46) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL8505150 0.94 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL8505677 0.86 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL8505563 0.82 PTGS2 (0.50) ALDH1A1KMT2AHPGDCYP2C9CYP2C19
SCHEMBL8506102 0.81 POLB (0.44) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL8502413 0.81 POLB (0.44) ALDH1A1MAPTLMNAHTTHPGD
Benzenesulfonamide SCHEMBL8525170 0.81 PTGS1 (0.44) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL8503362 0.77 ALDH1A1 (0.46) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL8504269 0.77 HTR6 (0.44) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL8503404 0.76 POLB (0.56) ALDH1A1MEN1KMT2AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP disclosed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO disclosed