SCHEMBL8525641

SCHEMBL8525641

N#Cc1ccc(CNC(=O)c2cccc3ccc(NS(=O)(=O)C4=CC=CN5SNC=C45)cc23)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATIC P31939 1/20 0.35
PPARA Q07869 1/20 0.35
KLKB1 P03952 2/20 0.34
KLK1 P06870 2/20 0.34
ELANE P08246 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
CNR2 P34972 2/20 0.33
NAMPT P43490 1/20 0.33
MCL1 Q07820 1/20 0.33
FNTA P49354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8523993 0.84 F10 (0.38) KLKB1HDAC2HDAC3HDAC4HDAC1
SCHEMBL8525755 0.73 HSP90AA1 (0.49) PPARACNR2MCL1AKR1B1
SCHEMBL8524454 0.72 PKLR (0.49) HDAC1
SCHEMBL1110102 0.69 TUBB (0.46) ATICPPARAKLKB1KLK1HDAC2
SCHEMBL3901212 0.69 CCKBR (0.42) GPR27
SCHEMBL3902502 0.68 CCKBR (0.34) ROCK2
SCHEMBL8525044 0.67 PKLR (0.49) HDAC1
SCHEMBL3900087 0.67 ALDH1A1 (0.43) ROCK2
SCHEMBL3910046 0.66 CCKBR (0.39) GPR27
SCHEMBL3900098 0.66 MEN1 (0.40) MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed