SCHEMBL8528932

SCHEMBL8528932

N#Cc1c(C(=O)O)ccc(-c2ccccc2)c1S(N)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.40
SLC22A12 Q96S37 2/20 0.40
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HNF4A P41235 2/20 0.37
ACMSD Q8TDX5 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
BIRC5 O15392 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533251 0.86 KDM4E (0.47) XDHSLC22A12ALDH1A1LMNAKMT2A
SCHEMBL8533389 0.84 SLC9A1 (0.38) ALDH1A1LMNAKMT2AKDM4ECYP1A2
SCHEMBL8534063 0.78 CA1 (0.42) ALDH1A1LMNAKMT2AHNF4AACMSD
SCHEMBL29788088 0.76 AKR1C2 (0.41) XDHSLC22A12ALDH1A1KMT2AKDM4E
SCHEMBL30153392 0.75 HNF4A (0.56) ALDH1A1LMNAKMT2AKDM4EHPGD
SCHEMBL29226029 0.75 HNF4A (0.56) ALDH1A1LMNAKMT2AKDM4EHPGD
SCHEMBL27784391 0.75 ADORA1 (0.42) XDHALDH1A1LMNAKMT2AKDM4E
SCHEMBL8530215 0.74 MEN1 (0.39) ALDH1A1LMNAKMT2AKDM4ECYP1A2
SCHEMBL8533248 0.74 FOLH1 (0.39) ALDH1A1LMNAKMT2ACYP2C9SMN1; SMN2
SCHEMBL28153772 0.74 HNF4A (0.54) XDHSLC22A12ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699660-B1 Arylbenzoylguanidines MERCK PATENT GMBH (DE) 1998-10-28 EP disclosed
US-5807896-A Arylbenzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTING (DE) 1998-09-15 US disclosed
EP-0699660-A2 Arylbenzoylguanidines MERCK PATENT GmbH (DE) 1996-03-06 EP disclosed