SCHEMBL8533251

SCHEMBL8533251

CS(=O)(=O)c1c(-c2ccccc2)ccc(C(=O)O)c1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
ALDH1A1 P00352 4/20 0.47
KMT2A Q03164 4/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
NPSR1 Q6W5P4 3/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.47
APAF1 O14727 1/20 0.41
USP2 O75604 1/20 0.41
PPARG P37231 1/20 0.41
NCOA2 Q15596 1/20 0.41
NCOA1 Q15788 1/20 0.41
GAA P10253 1/20 0.40
PAX8 Q06710 1/20 0.40
GRIA4 P48058 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528932 0.86 XDH (0.40) KDM4EALDH1A1KMT2ASMN1; SMN2NPSR1
SCHEMBL8529278 0.83 SLC9A1 (0.42) KDM4EALDH1A1KMT2ASMN1; SMN2NPSR1
SCHEMBL8529538 0.78 PTGS2 (0.41) KMT2ALMNAHPGDCYP1A2CYP2C9
SCHEMBL29788088 0.76 AKR1C2 (0.41) KDM4EALDH1A1KMT2ASMN1; SMN2GRIA4
SCHEMBL8529462 0.75 FOLH1 (0.40) ALDH1A1SMN1; SMN2PTGS2HNF4AFOLH1
SCHEMBL8529625 0.74 PTGS2 (0.38) KDM4EALDH1A1KMT2ASMN1; SMN2LMNA
SCHEMBL28153772 0.74 HNF4A (0.54) KDM4EALDH1A1KMT2ASMN1; SMN2GAA
SCHEMBL8610258 0.74 PTGS2 (0.39) ALDH1A1SMN1; SMN2LMNAPTGS2
SCHEMBL16911507 0.73 HNF4A (0.58) KDM4EALDH1A1KMT2ASMN1; SMN2LMNA
SCHEMBL5026544 0.73 FOLH1 (0.43) KDM4EALDH1A1KMT2ASMN1; SMN2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699660-B1 Arylbenzoylguanidines MERCK PATENT GMBH (DE) 1998-10-28 EP disclosed
US-5807896-A Arylbenzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTING (DE) 1998-09-15 US disclosed
EP-0699660-A2 Arylbenzoylguanidines MERCK PATENT GmbH (DE) 1996-03-06 EP disclosed