SCHEMBL8529082

SCHEMBL8529082

COc1c(F)cc(-n2nnnc2C)cc1C=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.38
NOTUM Q6P988 1/20 0.36
LMNA P02545 3/20 0.35
ATM Q13315 1/20 0.34
PRKCQ Q04759 6/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
ALDH1A1 P00352 2/20 0.31
HTT P42858 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
GALR3 O60755 1/20 0.31
TSHR P16473 1/20 0.31
LRRK2 Q5S007 1/20 0.31
S1PR4 O95977 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
S1PR1 P21453 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530190 0.81 ERN1 (0.45) KCNN4NOTUMLMNA
SCHEMBL4205532 0.76 ATM (0.45) NOTUMLMNAATMCA12CA9
SCHEMBL4201299 0.73 ALDH1A1 (0.52) NOTUMLMNAATMCA12CA9
SCHEMBL13743012 0.72 NOTUM (0.47) KCNN4NOTUMLMNACA12CA9
SCHEMBL8534986 0.70 CA1 (0.45) KCNN4LMNAATMALDH1A1HTT
SCHEMBL11041903 0.70 ERN1 (0.49) ALDH1A1TSHRKMT2ANPSR1SRC
SCHEMBL3814197 0.70 LMNA (0.47) KCNN4NOTUMLMNACA12CA9
SCHEMBL3823337 0.69 NOTUM (0.42) KCNN4NOTUMLMNAATMCA12
SCHEMBL13742929 0.69 NOTUM (0.47) KCNN4NOTUMLMNACA12CA9
SCHEMBL1186103 0.68 ERN1 (0.52) ALDH1A1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843966-A Piperidine derivatives GLAXO GROUP LIMITED (GB) 1998-12-01 US disclosed
EP-0720609-B1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LTD (GB) 1998-11-11 EP disclosed
US-5703240-A ANALGESICS; ANTIINFLAMMATORY AGENTS; NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS; GASTROINTESTINAL DISORDERS GLAXO GROUP LIMITED (GB) 1997-12-30 US disclosed
EP-0720609-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1996-07-10 EP disclosed
WO-1995008549-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1995-03-30 WO disclosed