SCHEMBL8529948

SCHEMBL8529948

O=C(O)C(CC(CCc1cccnc1)(C(=O)O)P(=O)(O)O)P(=O)(O)O

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FDPS P14324 7/20 0.55
BTN3A1 O00481 1/20 0.45
PDE3A Q14432 1/20 0.45
ANPEP P15144 2/20 0.43
ERAP2 Q6P179 1/20 0.43
ERAP1 Q9NZ08 1/20 0.43
TBXAS1 P24557 7/20 0.42
KDM4E B2RXH2 1/20 0.42
NAPRT Q6XQN6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532197 0.87 ANPEP (0.41) FDPSANPEPERAP2ERAP1
SCHEMBL8533589 0.85 FDPS (0.40) FDPSANPEPERAP2ERAP1
SCHEMBL8532177 0.79 FFAR1 (0.34)
SCHEMBL8530904 0.77 CYP1A2 (0.45) FDPS
SCHEMBL8528147 0.77 FDPS (0.46) FDPSANPEPERAP2ERAP1
SCHEMBL8745040 0.76 CYP2C19 (0.34) FDPSANPEPERAP2ERAP1KDM4E
SCHEMBL7863043 0.75 FDPS (0.69) FDPSBTN3A1PDE3AANPEPERAP2
SCHEMBL8532194 0.73 FDPS (0.45) FDPSBTN3A1PDE3AKDM4E
SCHEMBL8529344 0.72 FDPS (0.44) FDPSTBXAS1KDM4E
SCHEMBL8710665 0.72 FDPS (1.00) FDPSBTN3A1PDE3ATBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752999-B1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1998-10-28 EP disclosed
US-5698541-A DISEASES OF CALCIUM METABOLISM; OSTEOPOROSIS BOEHRINGER MANNHEIM GMBH (DE) 1997-12-16 US disclosed
EP-0752999-A1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM Roche Diagnostics GmbH (DE) 1997-01-15 EP disclosed
WO-1995026358-A1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1995-10-05 WO disclosed