SCHEMBL8530904

SCHEMBL8530904

O=C(O)C(CC(CCc1ccccn1)(C(=O)O)P(=O)(O)O)P(=O)(O)O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
FDPS P14324 2/20 0.45
PTPRA P18433 1/20 0.42
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.35
KCNA5 P22460 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532197 0.83 ANPEP (0.41) FDPS
SCHEMBL8533589 0.79 FDPS (0.40) FDPSSMN1; SMN2RAB9AALDH1A1HTT
SCHEMBL8529948 0.77 FDPS (0.55) FDPS
SCHEMBL8529344 0.76 FDPS (0.44) FDPSSMN1; SMN2HTT
SCHEMBL8532177 0.75 FFAR1 (0.34) SMN1; SMN2RAB9AL3MBTL1ALDH1A1
SCHEMBL8528147 0.75 FDPS (0.46) FDPSSMN1; SMN2
SCHEMBL8531643 0.71 FOLH1 (0.38) FDPS
SCHEMBL10622087 0.71 FDPS (0.71) CYP1A2FDPSCYP2C19SMN1; SMN2ALDH1A1
SCHEMBL9116044 0.71 FDPS (0.51) CYP1A2FDPSPTPRACYP2C19SMN1; SMN2
SCHEMBL7206606 0.71 CYP1A2 (0.56) CYP1A2FDPSPTPRACYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752999-B1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1998-10-28 EP disclosed
US-5698541-A DISEASES OF CALCIUM METABOLISM; OSTEOPOROSIS BOEHRINGER MANNHEIM GMBH (DE) 1997-12-16 US disclosed
EP-0752999-A1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM Roche Diagnostics GmbH (DE) 1997-01-15 EP disclosed
WO-1995026358-A1 2,4-DIPHOSPHONOGLUTARIC ACID DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1995-10-05 WO disclosed