SCHEMBL8533828

SCHEMBL8533828

CC(=O)O[C@@H]1NC(=O)[C@H]1NC(=O)[C@H](Cc1ccccc1)NS(=O)(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
MAPT P10636 1/20 0.61
CTSL P07711 11/20 0.60
CTSK P43235 11/20 0.60
CTSS P25774 7/20 0.60
CTSB P07858 1/20 0.51
MMP2 P08253 6/20 0.45
MMP9 P14780 6/20 0.45
ADAMTS4 O75173 1/20 0.45
MEN1 O00255 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449155 0.86 CTSL (0.60) ALDH1A1CTSLCTSKCTSSCTSB
SCHEMBL8086163 0.79 CTSK (0.79) CTSLCTSKCTSSCTSB
SCHEMBL31086837 0.77 ALDH1A1 (1.00) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL31086912 0.77 ALDH1A1 (0.80) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL7436896 0.76 CTSK (0.67) CTSLCTSKCTSSCTSB
SCHEMBL7160147 0.75 CTSK (1.00) CTSLCTSKCTSSCTSB
SCHEMBL7161878 0.75 CTSK (0.72) CTSLCTSKCTSSCTSB
SCHEMBL8086228 0.74 CTSK (0.49) CTSLCTSKCTSSCTSB
SCHEMBL8533829 0.74 ALDH1A1 (0.61) ALDH1A1MAPTMMP2MMP9ADAMTS4
SCHEMBL6021046 0.73 ALDH1A1 (0.73) ALDH1A1MAPTCTSLCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5986108-A ENZYME INHIBITORS SYNPHAR LABORATORIES, INC. (CA) 1999-11-16 US disclosed