SCHEMBL8534159

SCHEMBL8534159

CC(N)c1ccc(P(c2ccc(C(C)N)cc2)c2ccc(C(C)N)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.54
PDE2A O00408 1/20 0.43
TDP1 Q9NUW8 5/20 0.35
CYP3A4 P08684 1/20 0.35
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
CIT O14578 1/20 0.33
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
RECQL P46063 4/20 0.30
KDM4E B2RXH2 4/20 0.30
MAPT P10636 3/20 0.30
LMNA P02545 3/20 0.30
HIF1A Q16665 2/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
NFKB1 P19838 1/20 0.30
THPO P40225 1/20 0.30
HSD17B10 Q99714 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1314596 0.83 ADRB2 (0.72) ADRB2PDE2ATDP1ROCK2ROCK1
SCHEMBL3769642 0.78 TYR (0.44) ADRB2TDP1CYP3A4ESR1ESR2
SCHEMBL17540834 0.75 ADRB2 (0.70) ADRB2PDE2AKDM4EMAPTLMNA
SCHEMBL2187080 0.75 ADRB2 (0.70) ADRB2PDE2AKDM4EMAPTLMNA
SCHEMBL17540836 0.75 ADRB2 (0.70) ADRB2PDE2AKDM4EMAPTLMNA
SCHEMBL8535317 0.73 SLC6A4 (0.55) TDP1CYP3A4ESR1KDM4EMAPT
SCHEMBL334558 0.72 ADRB2 (0.59) ADRB2PDE2ATDP1LMNA
SCHEMBL353336 0.72 ADRB2 (0.59) ADRB2PDE2ATDP1LMNA
SCHEMBL342044 0.72 ADRB2 (0.59) ADRB2PDE2ATDP1CYP3A4ROCK2
Hydrochloric Acid SCHEMBL28673897 0.72 ADRB2 (0.67) ADRB2PDE2AROCK2ROCK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0789551-A4 HAIR CARE PERMING AGENTS AND PROCESSES LAU JOHN R (US) 1998-12-02 EP claimed
EP-0789551-A1 HAIR CARE PERMING AGENTS AND PROCESSES LAU, John R. (US) 1997-08-20 EP claimed
WO-1997011672-A1 HAIR CARE PERMING AGENTS AND PROCESSES LAU JOHN R (US) 1997-04-03 WO claimed