SCHEMBL8534293

SCHEMBL8534293

C=CCOc1ccc(C=O)cc1CC=C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
PTGDR Q13258 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.44
ALDH1A1 P00352 7/20 0.43
MAPT P10636 4/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
POLB P06746 2/20 0.41
FDPS P14324 1/20 0.41
MAPK1 P28482 1/20 0.41
TSHR P16473 2/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771880 0.84 ALDH1A1 (0.43) KDM4EALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL3464451 0.83 FDPS (0.54) KDM4EALDH1A1MAPTL3MBTL1LMNA
SCHEMBL4985231 0.82 ALDH1A1 (0.58) KDM4EALDH1A1MAPTL3MBTL1CYP1A2
SCHEMBL8416710 0.82 FDPS (0.44) KDM4EPTGDRPTGDR2ALDH1A1MAPT
SCHEMBL19251015 0.82 MAOA (0.46) ALDH1A1MAPTFDPSTSHRGAA
SCHEMBL5883140 0.81 MAOA (0.55) KDM4EPTGDRPTGDR2ALDH1A1MAPT
SCHEMBL5931990 0.80 GABRA1 (0.52) PTGDRPTGDR2MAPK1TSHRGAA
SCHEMBL4617044 0.79 TSHR (0.44) KDM4EALDH1A1MAPTLMNAFDPS
SCHEMBL31247739 0.79 FDPS (0.42) KDM4EALDH1A1MAPTTDP1FDPS
SCHEMBL18095839 0.79 ALDH1A1 (0.49) KDM4EALDH1A1POLBFDPSTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117624047-B Antitumor compound Beijing Keyou Ai Technology Co.,Ltd. (CN) 2026-05-26 CN disclosed
CN-117624048-A Antitumor nitrogen heterocyclic hydrazide compound 北京科佑爱科技有限责任公司 2024-03-01 CN disclosed
CN-117624047-A Antitumor compound 北京科佑爱科技有限责任公司 2024-03-01 CN disclosed
EP-0434394-B1 Compounds for treating inflammatory bowel disease LILLY CO ELI (US) 1998-08-05 EP disclosed
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed
US-5691367-A ANTIINFLAMMATORY AGENTS OR ANTIARTHRITIC AGENTS ELI LILLY AND COMPANY (US) 1997-11-25 US disclosed
WO-1996022772-A1 METHOD FOR TREATING MULTIPLE SCLEROSIS ELI LILLY AND COMPANY (US) 1996-08-01 WO disclosed
EP-0722729-A2 Aryl-substituted rhodanines for treating multiple sclerosis ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed
US-5387690-A Method of treating inflammatory bowel disease ELI LILLY AND COMPANY (US) 1995-02-07 US disclosed
US-5356917-A Antiischemic, antiinflammatory, antiarthritic agents, treat-ment of dystrophic mammals ELI LILLY AND COMPANY (US) 1994-10-18 US disclosed
US-5216002-A Using benzyl substituted rhodanine derivatives as pure enantiomeric form ELI LILLY AND COMPANY (US) 1993-06-01 US disclosed
US-5158966-A Aryl-substituted rhodanine derivatives THE UNIVERSITY OF COLORADO FOUNDATION, INC. (US) 1992-10-27 US disclosed
EP-0500337-A1 Composition containing aryl-substituted rhodanine derivatives for the treatment of type I diabetes UNIVERSITY OF COLORADO FOUNDATION, INC. (US) 1992-08-26 EP disclosed
EP-0434394-A2 Compounds for treating inflammatory bowel disease ELI LILLY AND COMPANY (US) 1991-06-26 EP disclosed