SCHEMBL8536502

SCHEMBL8536502

Cc1c(-c2cnn(Cc3ccc(OC(F)(F)F)cc3)c2)[nH]c2ccc(Cl)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.43
DDR1 Q08345 1/20 0.40
KLKB1 P03952 2/20 0.40
CHRM5 P08912 1/20 0.40
CNR1 P21554 2/20 0.38
KCNH2 Q12809 2/20 0.38
TYMS P04818 1/20 0.38
CYP3A4 P08684 1/20 0.38
GPR183 P32249 1/20 0.37
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
CREBBP Q92793 1/20 0.37
MARK4 Q96L34 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533234 0.93 MAT2A (0.49) MAT2ADDR1KLKB1CHRM5KCNH2
SCHEMBL8537370 0.91 MAT2A (0.43) MAT2AKLKB1CHRM5KCNH2TYMS
SCHEMBL8513871 0.89 MAT2A (0.46) MAT2AKLKB1CHRM5KCNH2TYMS
SCHEMBL8538579 0.85 MAT2A (0.61) MAT2AKLKB1CHRM5KCNH2TYMS
SCHEMBL8653277 0.85 MAT2A (0.49) MAT2AKLKB1CHRM5KCNH2TYMS
SCHEMBL8535741 0.80 ABL1 (0.41) KLKB1CHRM5KCNH2ABL1BCR
SCHEMBL9607468 0.80 MAT2A (0.44) MAT2ADDR1CNR1
SCHEMBL19002091 0.80 MAT2A (0.44) MAT2ACHRM5KCNH2ABL1ADORA2A
SCHEMBL8537111 0.79 MAT2A (0.55) MAT2ADDR1CNR1MEN1KMT2A
SCHEMBL8531391 0.78 CREBBP (0.40) KLKB1CHRM5KCNH2ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed