SCHEMBL8538579

SCHEMBL8538579

COc1ccc2c(=O)c(C)c(-c3cnn(Cc4ccc(OC(F)(F)F)cc4)c3)[nH]c2c1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.61
CYP19A1 P11511 4/20 0.41
ADORA2A P29274 2/20 0.40
ADORA2B P29275 2/20 0.40
ADORA1 P30542 2/20 0.40
KLKB1 P03952 2/20 0.40
CHRM5 P08912 4/20 0.39
KCNH2 Q12809 2/20 0.38
TYMS P04818 1/20 0.38
MGAT2 Q10469 1/20 0.37
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533234 0.91 MAT2A (0.49) MAT2ACYP19A1ADORA2AADORA2BADORA1
SCHEMBL8653277 0.91 MAT2A (0.49) MAT2ACYP19A1ADORA2AADORA2BADORA1
SCHEMBL8513871 0.89 MAT2A (0.46) MAT2AADORA2AADORA2BADORA1KLKB1
SCHEMBL8536502 0.85 MAT2A (0.43) MAT2AADORA2AADORA2BADORA1KLKB1
SCHEMBL8537370 0.85 MAT2A (0.43) MAT2AADORA2AADORA2BADORA1KLKB1
SCHEMBL8534140 0.84 ALDH1A1 (0.45) MAT2ACYP19A1ADORA2AADORA2BADORA1
SCHEMBL19002091 0.80 MAT2A (0.44) MAT2AADORA2AADORA2BADORA1CHRM5
SCHEMBL8537832 0.79 MAT2A (0.69) MAT2ACYP19A1
SCHEMBL8535741 0.78 ABL1 (0.41) ADORA2AADORA2BADORA1KLKB1CHRM5
SCHEMBL8530848 0.78 MAT2A (0.77) MAT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed