SCHEMBL8536754

SCHEMBL8536754

CC(C)Oc1ccc(-c2ccnc(N3CCN(CCN)CC3)n2)cc1C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 2/20 0.40
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
PIK3C3 Q8NEB9 1/20 0.39
KMO O15229 1/20 0.38
AAK1 Q2M2I8 3/20 0.36
SORD Q00796 1/20 0.36
HRH3 Q9Y5N1 3/20 0.35
PIK3CA P42336 1/20 0.34
ACHE P22303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515288 0.94 CARM1 (0.39) DKK1CTSSCTSKPIK3C3KMO
SCHEMBL8515329 0.91 ACHE (0.41) DKK1CTSSCTSKKMOSORD
SCHEMBL9612650 0.89 CARM1 (0.41) DKK1CTSSCTSKKMOSORD
SCHEMBL8510840 0.85 KMO (0.43) DKK1KMOSORDPIK3CA
SCHEMBL8511678 0.85 DKK1 (0.58) DKK1KMOAAK1SORDPIK3CA
SCHEMBL8515556 0.85 MEN1 (0.40) DKK1CTSSCTSKKMOSORD
SCHEMBL8512439 0.83 DKK1 (0.56) DKK1KMOSORDPIK3CA
SCHEMBL8511790 0.83 ROCK2 (0.41) DKK1KMOPIK3CAACHE
SCHEMBL8514120 0.83 KMO (0.40) DKK1KMOSORDPIK3CA
SCHEMBL8510713 0.83 KMO (0.39) DKK1KMOSORDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed