SCHEMBL9612650

SCHEMBL9612650

CC(C)Oc1ccc(-c2ccnc(N3CCN(CCN(C)C)CC3)n2)cc1C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.41
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
KMO O15229 1/20 0.37
RAD52 P43351 1/20 0.36
BRD4 O60885 3/20 0.36
MAPK14 Q16539 2/20 0.36
RPS6KB1 P23443 1/20 0.35
AKT1 P31749 1/20 0.35
DKK1 O94907 2/20 0.35
SORD Q00796 1/20 0.35
HRH3 Q9Y5N1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515288 0.96 CARM1 (0.39) CARM1CTSSCTSKKMORAD52
SCHEMBL8536754 0.89 DKK1 (0.40) CTSSCTSKKMODKK1SORD
SCHEMBL8515329 0.89 ACHE (0.41) CTSSCTSKKMODKK1SORD
SCHEMBL8510840 0.83 KMO (0.43) KMODKK1SORD
SCHEMBL8515556 0.83 MEN1 (0.40) CTSSCTSKKMODKK1SORD
SCHEMBL8515286 0.83 USP2 (0.35) CTSSCTSKKMODKK1SORD
SCHEMBL8511790 0.82 ROCK2 (0.41) KMODKK1
Hydrochloric Acid SCHEMBL8512525 0.81 ROCK2 (0.41) KMODKK1
SCHEMBL8514539 0.81 KMO (0.45) CTSSCTSKKMODKK1SORD
SCHEMBL8510671 0.81 DKK1 (0.44) KMODKK1SORD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed