SCHEMBL8536863

SCHEMBL8536863

NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)C(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.49
ERAP2 Q6P179 1/20 0.46
ERAP1 Q9NZ08 1/20 0.46
LNPEP Q9UIQ6 1/20 0.46
OPRD1 P41143 1/20 0.44
F2 P00734 3/20 0.43
ACE P12821 1/20 0.43
RAB9A P51151 1/20 0.42
SPHK2 Q9NRA0 1/20 0.42
SPHK1 Q9NYA1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13570514 0.86 F2 (0.53) DPP4ERAP2ERAP1LNPEPF2
SCHEMBL31376320 0.86 DPP4 (0.65) DPP4ERAP2ERAP1LNPEPF2
SCHEMBL6980126 0.85 AGTR2 (0.52) DPP4
SCHEMBL28797928 0.80 ERAP2 (0.48) DPP4ERAP2ERAP1LNPEPF2
SCHEMBL3733552 0.80 LMNA (0.52) DPP4ERAP2ERAP1LNPEPACE
SCHEMBL21067671 0.80 FKBP1A (0.51) OPRD1F2
SCHEMBL2176481 0.79 KCNH2 (0.47) DPP4ERAP2ERAP1LNPEPACE
SCHEMBL13570391 0.79 ERAP2 (0.45) DPP4ERAP2ERAP1LNPEPF2
SCHEMBL27828766 0.79 GAA (0.54) DPP4ERAP2ERAP1LNPEPACE
SCHEMBL17220302 0.79 GAA (0.54) DPP4ERAP2ERAP1LNPEPACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5714485-A Piperidine and hexahydropyridazine thrombin inhibitors MERCK & CO., INC. (US) 1998-02-03 US disclosed