SCHEMBL8537593

SCHEMBL8537593

O=[N+]([O-])c1cc(Cl)ccc1-c1ncc[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.47
CCNB2 O95067 1/20 0.47
CDK1 P06493 1/20 0.47
CCNB1 P14635 1/20 0.47
GSK3A P49840 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47
RAB9A P51151 3/20 0.46
MAPK1 P28482 4/20 0.45
TSHR P16473 1/20 0.45
NPC1 O15118 2/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
PDE7A Q13946 4/20 0.44
POLB P06746 2/20 0.44
PDE4B Q07343 1/20 0.43
PDE4D Q08499 1/20 0.43
PDE7B Q9NP56 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8541143 0.90 MAPK1 (0.51) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL5249670 0.83 MAPT (0.56) GSK3BRAB9AMAPK1TSHRNPC1
SCHEMBL8536034 0.82 ESR1 (0.43) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL8540810 0.82 TSHR (0.50) RAB9ATSHRNPC1MAPTNFKB1
SCHEMBL5528175 0.82 S100A4 (0.46) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL10680334 0.81 MAPT (0.39) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL1303527 0.80 CSNK1A1 (0.50) RAB9AMAPTHPGDALDH1A1L3MBTL1
SCHEMBL8536429 0.78 VCAM1 (0.50) MAPK1MAPTPDE4BPDE4DVCAM1
SCHEMBL8536432 0.78 ALDH1A1 (0.48) GSK3BRAB9AMAPK1NPC1MAPT
SCHEMBL6125034 0.78 MAPK1 (0.63) RAB9AMAPK1TSHRNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed