SCHEMBL8537739

SCHEMBL8537739

COc1ccc(C(=O)CCCCCBr)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.56
NPC1 O15118 4/20 0.56
PKM P14618 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.53
LMNA P02545 2/20 0.53
HTT P42858 2/20 0.53
THRA P10827 1/20 0.51
THRB P10828 1/20 0.51
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
USP2 O75604 1/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAPT P10636 1/20 0.48
ALDH1A1 P00352 1/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC3 O15379 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7267209 0.89 MAPT (0.55) HTTKMT2AMEN1MAPTALDH1A1
SCHEMBL1442018 0.86 NPC1 (0.56) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL21480338 0.85 RAB9A (0.59) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL11552829 0.84 HTR2A (0.52) RAB9ANPC1PKMLMNATHRA
SCHEMBL8537570 0.84 THRB (0.48) RAB9ANPC1PKMHTTTHRA
SCHEMBL8571284 0.84 RAB9A (0.58) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL9114685 0.84 NPC1 (0.57) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL10788695 0.84 SMN1; SMN2 (0.61) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL15076021 0.84 THRA (0.61) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL14930210 0.84 PDE4B (0.62) RAB9ANPC1PKMSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750532-A TETRAHYDROPYRIMIDINE-2,4-DIONE DERIVATIVES, VIRICIDES, ANTIINFLAMMATORY AGENTS, PAF INHIBITORS SCHERING CORPORATION (US) 1998-05-12 US disclosed
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed