SCHEMBL8538117

SCHEMBL8538117

NC(=O)Oc1ccc2[nH]cc(CCCCBr)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HTR1D P28221 9/20 0.53
MPO P05164 2/20 0.52
HTR1B P28222 9/20 0.51
HTR1A P08908 7/20 0.51
MTNR1A P48039 2/20 0.51
MTNR1B P49286 1/20 0.51
SLC6A4 P31645 1/20 0.50
TSHR P16473 2/20 0.49
HTR2C P28335 2/20 0.49
HTR7 P34969 2/20 0.49
HTR6 P50406 2/20 0.49
MEN1 O00255 1/20 0.49
HTR5A P47898 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2D6 P10635 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539513 0.89 CYP1A2 (0.64) CYP1A2CYP2C9CYP2C19HTR1DMPO
SCHEMBL10646261 0.89 HTR1D (0.57) CYP1A2CYP2C9CYP2C19HTR1DMPO
SCHEMBL9828421 0.89 HTR1D (0.67) CYP1A2CYP2C9CYP2C19HTR1DMPO
SCHEMBL8538858 0.88 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTR1DMPO
SCHEMBL9698903 0.85 MTNR1A (0.56) CYP1A2CYP2C9CYP2C19HTR1DMPO
SCHEMBL10557687 0.84 CYP1A2 (0.76) CYP1A2CYP2C9CYP2C19HTR1DHTR1B
SCHEMBL9264998 0.82 HTR7 (0.72) CYP1A2CYP2C9HTR1DMPOHTR1B
SCHEMBL8538964 0.82 HTR1A (0.48) CYP1A2CYP2C9CYP2C19HTR1DHTR1B
SCHEMBL9329223 0.80 SLC6A4 (0.69) CYP1A2CYP2C9HTR1DHTR1BHTR1A
SCHEMBL9827891 0.79 HTR1D (0.67) CYP1A2CYP2C9CYP2C19HTR1DMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496222-B1 Indole derivatives MERCK PATENT GMBH (DE) 1998-09-09 EP disclosed
EP-0496222-A1 Indole derivatives MERCK PATENT GmbH (DE) 1992-07-29 EP disclosed