SCHEMBL8538964

SCHEMBL8538964

O=C(Oc1ccc2[nH]cc(CCCCBr)c2c1)N1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.48
HTR1D P28221 5/20 0.48
HTR1B P28222 5/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTR2A P28223 2/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544087 0.88 HTR1D (0.50) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL10646261 0.83 HTR1D (0.57) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL9828421 0.83 HTR1D (0.67) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL9258017 0.82 HRH3 (0.55) HTR1AHTR1DHTR1BCYP1A2ALDH1A1
SCHEMBL8538117 0.82 CYP1A2 (0.56) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL8539020 0.81 ADRA2A (0.62)
SCHEMBL8543448 0.80 ADRA2A (0.61)
SCHEMBL9698903 0.80 MTNR1A (0.56) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL9329223 0.75 SLC6A4 (0.69) HTR1AHTR1DHTR1BCYP1A2CYP2C9
SCHEMBL12720724 0.73 MTNR1A (0.52) HTR1ACYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496222-B1 Indole derivatives MERCK PATENT GMBH (DE) 1998-09-09 EP disclosed
EP-0496222-A1 Indole derivatives MERCK PATENT GmbH (DE) 1992-07-29 EP disclosed