SCHEMBL8539455

SCHEMBL8539455

Cc1ccc(S(=O)(=O)OCCC(CC(=O)O)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.48
CASP1 P29466 2/20 0.47
LMNA P02545 1/20 0.46
CTRB1 P17538 2/20 0.46
CASP3 P42574 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539453 1.00 P2RX7 (0.48) P2RX7CASP1LMNACTRB1CASP3
SCHEMBL3070245 0.83 P2RX7 (0.48) P2RX7LMNACTRB1CA1CA2
SCHEMBL9476901 0.83 CTRB1 (0.56) P2RX7LMNACTRB1CA1CA2
SCHEMBL7990292 0.81 LMNA (0.48) P2RX7LMNACTRB1CA1CA2
SCHEMBL3652008 0.80 P2RX7 (0.51) P2RX7LMNACA1CA2MAPT
SCHEMBL3652010 0.80 P2RX7 (0.51) P2RX7LMNACA1CA2MAPT
SCHEMBL22552853 0.80 P2RX7 (0.51) P2RX7LMNACA1CA2MAPT
SCHEMBL6924285 0.80 LMNA (0.59) P2RX7LMNACA1CA2MAPT
SCHEMBL7990303 0.79 P2RX7 (0.47) P2RX7LMNACTRB1CA1CA2
SCHEMBL3957822 0.79 P2RX7 (0.54) P2RX7CASP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0565396-B1 1-[2-(arylsulfonylamino)-1-oxoethyl]piperidine derivatives, their preparation and use in therapy SYNTHELABO (FR) 1998-01-07 EP disclosed
EP-0579277-A1 Imidazole derivatives, their preparation and their use as synthetic intermediates SYNTHELABO (FR) 1994-01-19 EP disclosed