SCHEMBL8540658

SCHEMBL8540658

CS(=O)(=O)Cc1cc(O)ccc1-c1ncc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.48
JAK1 P23458 2/20 0.48
TYK2 P29597 2/20 0.48
JAK3 P52333 2/20 0.48
ADRA1A P35348 2/20 0.39
CDK4 P11802 1/20 0.38
CCNA2 P20248 1/20 0.38
CCND1 P24385 1/20 0.38
CDK2 P24941 1/20 0.38
CCND3 P30281 1/20 0.38
CSNK1A1 P48729 1/20 0.38
TYRO3 Q06418 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
CASP6 P55212 1/20 0.36
SMPD3 Q9NY59 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NISCH Q9Y2I1 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540682 0.84 CSNK1A1 (0.47) JAK2JAK1TYK2JAK3ADRA1A
SCHEMBL8539349 0.80 HCRTR1 (0.40) JAK2JAK1TYK2JAK3ADRA1A
SCHEMBL8536816 0.77 JAK2 (0.47) JAK2JAK1TYK2JAK3ADRA1A
SCHEMBL8538833 0.75 JAK2 (0.46) JAK2JAK1TYK2JAK3ADRA1A
SCHEMBL8537911 0.73 AMY1A (0.45) JAK2JAK1TYK2JAK3CDK4
SCHEMBL8536858 0.72 ESR2 (0.46) JAK2JAK1TYK2JAK3CDK4
SCHEMBL31429641 0.72 GUSB (0.45) JAK2JAK1TYK2JAK3CDK4
SCHEMBL8540911 0.72 GUSB (0.45) JAK2JAK1TYK2JAK3CDK4
SCHEMBL8613204 0.71 CSNK1A1 (0.46) JAK2JAK1TYK2JAK3ADRA1A
SCHEMBL31429688 0.71 CSNK1A1 (0.44) JAK2JAK1TYK2JAK3CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed