SCHEMBL8539349

SCHEMBL8539349

CS(=O)(=O)Cc1cc(C#N)ccc1-c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CYP19A1 P11511 2/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ADRA1A P35348 1/20 0.37
EGLN2 Q96KS0 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
ATR Q13535 1/20 0.34
SRPK2 P78362 1/20 0.33
SRPK1 Q96SB4 1/20 0.33
S100A9 P06702 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540658 0.80 JAK2 (0.48) ADRA1APDE4APDE4BPDE4CPDE4D
SCHEMBL8539601 0.79 CYP19A1 (0.41) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL8540682 0.78 CSNK1A1 (0.47) CYP19A1ADRA1ACSNK1A1TYRO3DYRK1B
SCHEMBL8541136 0.77 CYP19A1 (0.39) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL8535598 0.75 CYP19A1 (0.46) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL31486076 0.71 CYP19A1 (0.45) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL8536429 0.69 VCAM1 (0.50) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL8540558 0.68 VCAM1 (0.46) HCRTR1HCRTR2CYP19A1CYP11B1CYP11B2
SCHEMBL8617021 0.68 CSNK1A1 (0.44) ADRA1ACSNK1A1TYRO3DYRK1BNISCH
SCHEMBL22637167 0.67 MBOAT4 (0.41) CYP11B1CYP11B2TRPV4HRH4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed