SCHEMBL8540877

SCHEMBL8540877

Cc1ccc(S(=O)(=O)OC[C@@H]2CCN(Cc3ccccc3)C2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.52
BCHE P06276 2/20 0.50
LMNA P02545 3/20 0.49
ALDH1A1 P00352 2/20 0.49
TSHR P16473 1/20 0.49
ACHE P22303 2/20 0.49
BACE1 P56817 2/20 0.49
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
CD4 P01730 2/20 0.47
SORT1 Q99523 1/20 0.47
POLB P06746 1/20 0.47
OPRM1 P35372 1/20 0.46
OPRK1 P41145 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540875 1.00 HTR6 (0.54) HTR6SMN1; SMN2BCHELMNAALDH1A1
SCHEMBL1943416 0.93 ACHE (0.53) HTR6SMN1; SMN2BCHEACHECD4
SCHEMBL14166152 0.93 SMN1; SMN2 (0.56) HTR6SMN1; SMN2LMNAALDH1A1TSHR
SCHEMBL9212450 0.92 BCHE (0.50) HTR6SMN1; SMN2BCHELMNAALDH1A1
SCHEMBL9217317 0.91 HTR2A (0.55) HTR6BCHEALDH1A1ACHEDRD2
SCHEMBL19475540 0.88 SMN1; SMN2 (0.55) HTR6SMN1; SMN2LMNAALDH1A1TSHR
SCHEMBL7782471 0.88 HTR6 (0.53) HTR6SMN1; SMN2BCHELMNAALDH1A1
SCHEMBL1474769 0.84 SMN1; SMN2 (0.48) HTR6SMN1; SMN2BCHELMNAALDH1A1
SCHEMBL1474768 0.84 SMN1; SMN2 (0.48) HTR6SMN1; SMN2BCHELMNAALDH1A1
SCHEMBL1474765 0.84 SMN1; SMN2 (0.48) HTR6SMN1; SMN2BCHELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770611-A Indole derivatives as 5HT1 -like agonists PFIZER INC. (US) 1998-06-23 US disclosed
EP-0785933-B1 INDOLE DERIVATIVES AS 5HT1-LIKE AGONISTS PFIZER LTD (GB) 1998-03-11 EP disclosed
EP-0785933-A1 INDOLE DERIVATIVES AS 5HT1-LIKE AGONISTS Pfizer Limited (GB) 1997-07-30 EP disclosed
WO-1996011195-A1 INDOLE DERIVATIVES AS 5HT1-LIKE AGONISTS PFIZER LIMITED (GB) 1996-04-18 WO disclosed