SCHEMBL8540903

SCHEMBL8540903

CSc1ccc(C2=CCCC3CN(C)CC23)cc1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.33
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KCNH2 Q12809 1/20 0.31
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466006 0.82 HRH3 (0.42) HRH3
SCHEMBL15428837 0.68 SIGMAR1 (0.33) HRH3
SCHEMBL3058175 0.66 HRH3 (0.74) HRH3KCNH2
SCHEMBL23605127 0.65 PTGS2 (0.33) HRH3ALDH1A1HPGDHSD17B10
SCHEMBL14594807 0.64 SIGMAR1 (0.31)
SCHEMBL8539768 0.64 SLC6A4 (0.36) ALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL9530988 0.63 SLC18A3 (0.31) DRD2DRD4
SCHEMBL10300271 0.59 ALDH1A1 (0.50) ALDH1A1
SCHEMBL10528160 0.59 ALDH1A1 (0.50) ALDH1A1
SCHEMBL8967524 0.58 ALDH1A1 (0.32) ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690842-B1 4-ARYLISOINDOLE ANALGESICS ORTHO PHARMA CORP (US) 1998-12-16 EP disclosed
US-5508424-A REDUCED SIDE EFFECTS ORTHO PHARMACEUTICAL CORPORATION (US) 1996-04-16 US disclosed