SCHEMBL8544971

SCHEMBL8544971

c1ccc(CCCN2CCC(CCn3cnc(-c4ccccc4)c3-c3ccccc3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.51
GRIN2B Q13224 1/20 0.50
SIGMAR1 Q99720 3/20 0.49
CCR3 P51677 1/20 0.49
HRH3 Q9Y5N1 4/20 0.48
HTR2A P28223 1/20 0.46
KCNH2 Q12809 1/20 0.46
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037240 0.91 GRIN2B (0.45) ACHEGRIN2BSIGMAR1CCR3HRH3
SCHEMBL8541891 0.82 HTT (0.63) ACHEGRIN2BSIGMAR1CCR3HRH3
SCHEMBL8545141 0.81 PTGS2 (0.53) ACHEGRIN2B
SCHEMBL8696219 0.80 PTGS2 (0.43)
SCHEMBL8539516 0.80 HRH3 (0.53) ACHEGRIN2BSIGMAR1CCR3HRH3
SCHEMBL8539193 0.79 GRIN2B (0.54) GRIN2BSIGMAR1CCR3HRH3HTR2A
SCHEMBL83059 0.76 SIGMAR1 (0.69) GRIN2BSIGMAR1CCR3HRH3
SCHEMBL8540771 0.76 GRIN2B (0.58) GRIN2BSIGMAR1CCR3HRH3SLC6A4
SCHEMBL8542377 0.75 HRH3 (0.53) GRIN2BSIGMAR1CCR3HRH3
SCHEMBL8543286 0.75 GRIN2B (0.55) GRIN2BSIGMAR1CCR3HRH3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed