SCHEMBL8545141

SCHEMBL8545141

O=C(CCc1ccccc1)N1CCC(CCn2cnc(-c3ccccc3)c2-c2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.53
FAAH O00519 2/20 0.53
GRIN2B Q13224 1/20 0.52
POLB P06746 1/20 0.50
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA4 P43681 1/20 0.48
CPB1 P15086 1/20 0.48
NPC1 O15118 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NAAA Q02083 1/20 0.46
ACHE P22303 1/20 0.45
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
FKBP1A P62942 1/20 0.44
TSHR P16473 1/20 0.43
YAP1 P46937 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542324 0.83 HTT (0.58) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8544549 0.81 GRIN2B (0.53) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8702971 0.81 PTGS2 (0.50) PTGS2NPC1TDP1NAAA
SCHEMBL8544971 0.81 ACHE (0.51) GRIN2BACHE
SCHEMBL8541896 0.80 FAAH (0.56) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8544779 0.78 GRIN2B (0.60) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8545115 0.77 POLB (0.52) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8546968 0.77 F10 (0.57) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8539166 0.76 GRIN2B (0.54) FAAHGRIN2BPOLBCHRNB2CHRNB4
SCHEMBL8545014 0.75 CPB1 (0.60) FAAHGRIN2BPOLBCHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed