SCHEMBL8545219

SCHEMBL8545219

O=C(NCc1ccccc1)[C@@H]1CCCN1CC(=O)C1(c2ccc(Cl)cc2)CCCCC1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 1/20 0.54
POLB P06746 2/20 0.50
CACNA1G O43497 1/20 0.49
F2 P00734 4/20 0.49
FKBP1A P62942 1/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
PKM P14618 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
TRPA1 O75762 1/20 0.44
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550285 0.93 FKBP1A (0.49) EP300POLBCACNA1GF2FKBP1A
SCHEMBL8548639 0.90 CYP3A4 (0.57) EP300CACNA1GF2FKBP1AALDH1A1
SCHEMBL8545217 0.85 EP300 (0.48) EP300CACNA1GHSD11B1
SCHEMBL8545214 0.85 EP300 (0.48) EP300CACNA1GHSD11B1
SCHEMBL8549405 0.82 CYP3A4 (0.52) POLBCACNA1GF2FKBP1AALDH1A1
SCHEMBL8543073 0.81 F2 (0.56) POLBF2FKBP1AALDH1A1CYP3A4
SCHEMBL8544795 0.78 FKBP1A (0.59) POLBF2FKBP1AALDH1A1CYP3A4
SCHEMBL8550278 0.77 EP300 (0.42) EP300CACNA1GSMN1; SMN2
SCHEMBL8550282 0.77 EP300 (0.42) EP300CACNA1GSMN1; SMN2
SCHEMBL7452551 0.76 FKBP1A (0.60) POLBCACNA1GF2FKBP1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed