SCHEMBL8550285

SCHEMBL8550285

O=C(NCc1ccccc1)[C@@H]1CCCN1CC(=O)C1(c2ccccc2)CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 2/20 0.49
CACNA1G O43497 1/20 0.48
ALDH1A1 P00352 4/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
EP300 Q09472 1/20 0.47
F2 P00734 2/20 0.47
POLB P06746 1/20 0.46
PTGER4 P35408 2/20 0.46
USP2 O75604 1/20 0.44
HPGD P15428 1/20 0.44
ERCC1 P07992 1/20 0.44
ERCC4 Q92889 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545219 0.93 EP300 (0.54) FKBP1ACACNA1GALDH1A1CYP3A4CYP2C9
SCHEMBL8548639 0.93 CYP3A4 (0.57) FKBP1ACACNA1GALDH1A1CYP3A4CYP2C9
SCHEMBL8549405 0.86 CYP3A4 (0.52) FKBP1ACACNA1GALDH1A1CYP3A4CYP2C9
SCHEMBL8550278 0.83 EP300 (0.42) CACNA1GSMN1; SMN2EP300
SCHEMBL8550282 0.83 EP300 (0.42) CACNA1GSMN1; SMN2EP300
SCHEMBL8544795 0.81 FKBP1A (0.59) FKBP1AALDH1A1CYP3A4CYP2C9PKM
SCHEMBL8544266 0.80 HPGD (0.54) FKBP1AALDH1A1CYP3A4CYP2C9PKM
SCHEMBL8543317 0.78 F2 (0.58) FKBP1AALDH1A1CYP3A4CYP2C9PKM
SCHEMBL7452551 0.78 FKBP1A (0.60) FKBP1ACACNA1GALDH1A1CYP3A4CYP2C9
SCHEMBL2441194 0.78 FKBP1A (0.60) FKBP1ACACNA1GALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed