SCHEMBL8549405

SCHEMBL8549405

CC1(C(=O)CN2CCC[C@H]2C(=O)NCc2ccccc2)CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
PKM P14618 1/20 0.52
CYP2C19 P33261 1/20 0.52
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
FKBP1A P62942 3/20 0.50
F2 P00734 4/20 0.48
CACNA1G O43497 1/20 0.47
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
PTGER4 P35408 2/20 0.46
AADAT Q8N5Z0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550285 0.86 FKBP1A (0.49) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8548639 0.84 CYP3A4 (0.57) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8549394 0.83 ACE (0.42) ALDH1A1SMN1; SMN2CACNA1GNPC1GAA
SCHEMBL8549403 0.83 ACE (0.42) ALDH1A1SMN1; SMN2CACNA1GNPC1GAA
SCHEMBL8544795 0.82 FKBP1A (0.59) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8545219 0.82 EP300 (0.54) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8545031 0.81 ALDH1A1 (0.61) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8544266 0.80 HPGD (0.54) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL8543317 0.79 F2 (0.58) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL7452551 0.79 FKBP1A (0.60) CYP3A4CYP2C9PKMCYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed