SCHEMBL8545352

SCHEMBL8545352

O=C(CN1CCC[C@@H]1C(=O)NC(=O)c1ccccc1)c1cccc(OC(=O)c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.43
CTSK P43235 8/20 0.42
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
MEN1 O00255 1/20 0.39
SPHK1 Q9NYA1 2/20 0.39
SPHK2 Q9NRA0 1/20 0.39
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545349 1.00 KMT2A (0.46) KMT2AALDH1A1MAPTCTSKCHRNB2
SCHEMBL8548486 0.90 CTSK (0.46) KMT2AALDH1A1MAPTCTSKMEN1
SCHEMBL8548482 0.90 CTSK (0.46) KMT2AALDH1A1MAPTCTSKMEN1
SCHEMBL8544653 0.90 ERCC5 (0.49) KMT2ACTSKMEN1RAB9A
SCHEMBL8544642 0.90 ERCC5 (0.49) KMT2ACTSKMEN1RAB9A
SCHEMBL8548133 0.89 MEN1 (0.51) KMT2AALDH1A1CTSKMEN1RAB9A
SCHEMBL8548127 0.89 MEN1 (0.51) KMT2AALDH1A1CTSKMEN1RAB9A
SCHEMBL8543631 0.86 SPHK1 (0.54) KMT2AALDH1A1MEN1SPHK1SPHK2
SCHEMBL8543635 0.86 SPHK1 (0.54) KMT2AALDH1A1MEN1SPHK1SPHK2
SCHEMBL8545355 0.86 ALDH1A1 (0.51) KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed