SCHEMBL8545520

SCHEMBL8545520

NC(=O)N(Cc1ccc(N)cc1)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIB P23284 1/20 0.51
PPID Q08752 1/20 0.51
PPIG Q13427 1/20 0.51
MAOB P27338 5/20 0.44
MAOA P21397 3/20 0.44
RAB9A P51151 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALOX5 P09917 3/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
F2 P00734 1/20 0.40
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40
NPC1 O15118 1/20 0.40
PARP10 Q53GL7 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320045 0.92 PARP10 (0.44) PPIBPPIDPPIGRAB9AL3MBTL1
SCHEMBL8550259 0.89 PLA2G10 (0.49) PPIBPPIDPPIGRAB9AL3MBTL1
SCHEMBL8545528 0.87 NR3C1 (0.48) L3MBTL1ALOX5PTGS1PTGS2PARP10
SCHEMBL8547009 0.87 NR3C1 (0.48) L3MBTL1ALOX5PTGS1PTGS2PARP10
SCHEMBL8549653 0.83 LPAR1 (0.46) L3MBTL1ALOX5PTGS1PTGS2
SCHEMBL8550313 0.83 MEN1 (0.49) RAB9AL3MBTL1SMN1; SMN2ALOX5PTGS1
SCHEMBL8551384 0.82 CRHBP (0.53) RAB9ASMN1; SMN2NPC1LMNAALDH1A1
SCHEMBL8546552 0.82 MEN1 (0.48) L3MBTL1ALOX5PTGS1PTGS2PARP10
SCHEMBL8546496 0.81 NR3C1 (0.47) ALOX5KDM4EALDH1A1
SCHEMBL8543702 0.81 ACHE (0.49) L3MBTL1SMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1045005-C Novel bisoxadiazolidine derivative YAMANOUCHI PHARMA CO LTD (JP) 1999-09-08 CN disclosed
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
CN-1122133-A Novel bis-oxadiazolidine derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-05-08 CN disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed