SCHEMBL8550259

SCHEMBL8550259

NC(=O)N(Cc1ccc(Cc2ccc(CN(OCc3ccccc3)C(N)=O)cc2)cc1)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.49
PLA2G2A P14555 1/20 0.49
ALOX5 P09917 3/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
LMNA P02545 1/20 0.41
PPIB P23284 1/20 0.41
PPID Q08752 1/20 0.41
PPIG Q13427 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
SLC22A2 O15244 1/20 0.40
PARP10 Q53GL7 1/20 0.40
LTA4H P09960 1/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PPARG P37231 3/20 0.38
PPARA Q07869 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320045 0.94 PARP10 (0.44) ALOX5PTGS1PTGS2PPIBPPID
SCHEMBL8545520 0.89 PPIB (0.51) ALOX5PTGS1PTGS2LMNAPPIB
SCHEMBL8547009 0.88 NR3C1 (0.48) ALOX5PTGS1PTGS2L3MBTL1PARP10
SCHEMBL8545528 0.88 NR3C1 (0.48) ALOX5PTGS1PTGS2L3MBTL1PARP10
SCHEMBL8550313 0.84 MEN1 (0.49) ALOX5PTGS1PTGS2L3MBTL1PARP10
SCHEMBL8549653 0.84 LPAR1 (0.46) ALOX5PTGS1PTGS2L3MBTL1
SCHEMBL8551384 0.83 CRHBP (0.53) LMNAALDH1A1NPC1RAB9A
SCHEMBL8546552 0.83 MEN1 (0.48) ALOX5PTGS1PTGS2L3MBTL1PARP10
SCHEMBL8546496 0.82 NR3C1 (0.47) ALOX5ALDH1A1
SCHEMBL8543702 0.82 ACHE (0.49) L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed