SCHEMBL8548156

SCHEMBL8548156

Fc1ccc(-c2nncc3c(C(F)(F)C(F)(F)F)cccc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ESR1 P03372 1/20 0.36
NR1H2 P55055 4/20 0.34
NR1H3 Q13133 4/20 0.34
NPSR1 Q6W5P4 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 3/20 0.33
LMNA P02545 1/20 0.33
ADORA2A P29274 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMO Q99835 1/20 0.33
ENPP1 P22413 1/20 0.33
NR1I2 O75469 1/20 0.32
NR3C1 P04150 1/20 0.32
EGFR P00533 1/20 0.32
KDR P35968 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28877285 0.70 EGFR (0.55) SMN1; SMN2ALDH1A1ESR1KDM4EMAPT
SCHEMBL8552083 0.70 MEN1 (0.34) SMN1; SMN2ALDH1A1ESR1NR1H2NR1H3
SCHEMBL8551923 0.69 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1NPSR1KDM4EMAPT
SCHEMBL8552079 0.68 SMN1; SMN2 (0.34) SMN1; SMN2ALDH1A1KDM4EMAPTLMNA
SCHEMBL8551133 0.66 NR1H2 (0.42) ESR1NR1H2NR1H3MAPTADORA2A
SCHEMBL1407266 0.63 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1NR1H2NR1H3KDM4E
SCHEMBL1268020 0.62 ESR1 (0.49) SMN1; SMN2ALDH1A1ESR1NPSR1MAPT
SCHEMBL14959329 0.62 KDM4E (0.56) SMN1; SMN2ALDH1A1ESR1NPSR1KDM4E
SCHEMBL18936152 0.61 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL15913865 0.61 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed