SCHEMBL8551133

SCHEMBL8551133

Fc1ccc(-c2nnc(Cl)c3c(C(F)(F)F)cccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 7/20 0.42
NR1H3 Q13133 7/20 0.42
NR1I2 O75469 2/20 0.40
NR3C1 P04150 2/20 0.40
AR P10275 1/20 0.40
RXRA P19793 1/20 0.40
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
P2RX7 Q99572 4/20 0.36
ESR1 P03372 3/20 0.36
MAPT P10636 1/20 0.36
ENPP1 P22413 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552718 0.89 ALDH1A1 (0.42) ESR1MAPTENPP1
SCHEMBL8546259 0.88 NR1H2 (0.41) NR1H2NR1H3ADORA2AADORA1ESR1
SCHEMBL8547763 0.79 ADORA2A (0.38) ADORA2AADORA1ESR1MAPT
SCHEMBL8551877 0.79 ESR1 (0.37) ADORA2AADORA1ESR1MAPT
SCHEMBL26614999 0.77 KDM4E (0.39) NR1H2NR1H3ENPP1
SCHEMBL8553715 0.77 NR1H2 (0.38) NR1H2NR1H3NR1I2NR3C1AR
SCHEMBL1268020 0.75 ESR1 (0.49) ADORA2AESR1MAPT
SCHEMBL8553708 0.75 LMNA (0.35) NR1H2NR1H3NR1I2NR3C1ADORA2A
SCHEMBL8551845 0.73 ROCK2 (0.48) NR1H2NR1H3ARP2RX7MAPT
SCHEMBL1407266 0.72 SMN1; SMN2 (0.50) NR1H2NR1H3NR1I2NR3C1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed