SCHEMBL8552079

SCHEMBL8552079

N=C(N)Nc1nnc(-c2ccc(F)cc2)c2cccc(C(F)(F)C(F)(F)F)c12

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 4/20 0.33
KDR P35968 6/20 0.32
ENPP3 O14638 1/20 0.32
THRB P10828 1/20 0.31
CA9 Q16790 1/20 0.31
KCNJ11 Q14654 1/20 0.31
GAA P10253 2/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 2/20 0.31
BRAF P15056 1/20 0.31
HTT P42858 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553708 0.91 LMNA (0.35) SMN1; SMN2LMNAMAPTKDRENPP3
SCHEMBL8551148 0.85 ENPP3 (0.38) SMN1; SMN2LMNAMAPTKDRENPP3
SCHEMBL8553998 0.81 KDR (0.37) SMN1; SMN2LMNAMAPTKDRENPP3
SCHEMBL8546406 0.81 SMN1; SMN2 (0.36) SMN1; SMN2LMNAMAPTKDRENPP3
SCHEMBL8550319 0.81 KDM4E (0.37) SMN1; SMN2MAPTKDRENPP3THRB
SCHEMBL8547661 0.81 ALDH1A1 (0.43) SMN1; SMN2MAPTKDRENPP3THRB
Hydrochloric Acid SCHEMBL8548628 0.81 KDM4E (0.37) SMN1; SMN2MAPTKDRENPP3THRB
SCHEMBL8552083 0.77 MEN1 (0.34) SMN1; SMN2LMNAMAPTALDH1A1POLB
SCHEMBL8374822 0.70 NPSR1 (0.39) SMN1; SMN2MAPTKDRENPP3THRB
SCHEMBL8518196 0.70 NPSR1 (0.39) SMN1; SMN2MAPTKDRENPP3THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed