SCHEMBL8548238

SCHEMBL8548238

COc1cc(C(Br)C(=O)c2ccccc2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 2/20 0.50
ATM Q13315 2/20 0.48
TNFRSF1A P19438 1/20 0.47
KMT2A Q03164 5/20 0.45
MEN1 O00255 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 2/20 0.44
THRB P10828 1/20 0.44
HTT P42858 1/20 0.44
MAPK1 P28482 1/20 0.44
ABCB1 P08183 1/20 0.43
TSHR P16473 1/20 0.43
CYP2D6 P10635 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11369147 0.85 NPC1 (0.49) ALDH1A1CYP1A2TNFRSF1ASMN1; SMN2MAPT
SCHEMBL2040575 0.83 CES2 (0.56) ALDH1A1CYP1A2ATMTNFRSF1AKMT2A
SCHEMBL9530939 0.78 ALDH1A1 (0.56) ALDH1A1CYP1A2ATMTNFRSF1AKMT2A
SCHEMBL11202653 0.77 HTT (0.46) ALDH1A1MAPTHTTMAPK1TSHR
SCHEMBL7017619 0.76 ALDH1A1 (0.57) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL11376411 0.76 CA12 (0.56) ALDH1A1CYP1A2TNFRSF1AKMT2AMEN1
SCHEMBL7146375 0.75 CYP1A2 (0.51) CYP1A2ABCB1CYP2C19
Bromide SCHEMBL6282375 0.74 CYP1A2 (0.50) CYP1A2ABCB1CYP2C19
SCHEMBL627867 0.74 CES2 (0.64) ALDH1A1ATMSMN1; SMN2HTTMAPK1
SCHEMBL2040577 0.74 LMNA (0.56) ALDH1A1CYP1A2TNFRSF1AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000014073-A1 BENZODIAZEPINONE DERIVATIVES, PREPARATION METHOD AND INTERMEDIATES THEREFOR, USE AS MEDICINES AND COMPOSITIONS HOECHST MARION ROUSSEL (FR) 2000-03-16 WO claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed