SCHEMBL8552718

SCHEMBL8552718

Cc1ccc(-c2nnc(Cl)c3c(C(F)(F)F)cccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
HTT P42858 5/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 5/20 0.40
NPSR1 Q6W5P4 6/20 0.39
LMNA P02545 4/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TRPV1 Q8NER1 1/20 0.38
HPGD P15428 1/20 0.37
ENPP1 P22413 1/20 0.37
ESR1 P03372 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551133 0.89 NR1H2 (0.42) MAPTENPP1ESR1
SCHEMBL8546259 0.88 NR1H2 (0.41) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL8550781 0.79 ALDH1A1 (0.44) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL8547668 0.78 PLAU (0.37) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL8547661 0.76 ALDH1A1 (0.43) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL8551333 0.76 ALDH1A1 (0.41) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL8548542 0.75 ROCK2 (0.47) ALDH1A1SMN1; SMN2MAPTNPSR1LMNA
SCHEMBL7904780 0.75 ALDH1A1 (0.60) ALDH1A1HTTSMN1; SMN2MAPTNPSR1
SCHEMBL26614999 0.74 KDM4E (0.39) SMN1; SMN2NPSR1KDM4ETRPV1ENPP1
SCHEMBL8548608 0.74 MAPT (0.44) ALDH1A1HTTSMN1; SMN2MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed