SCHEMBL8548715

SCHEMBL8548715

CCc1csc(C(O)C(=O)c2ccc(F)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
LMNA P02545 4/20 0.40
GAA P10253 2/20 0.39
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37
MAPT P10636 3/20 0.36
RAB9A P51151 1/20 0.36
HTR7 P34969 1/20 0.36
CNR2 P34972 1/20 0.35
HPGD P15428 2/20 0.35
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CES2 O00748 3/20 0.34
CES1 P23141 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HTT P42858 2/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087828 0.81 SMN1; SMN2 (0.37) ALDH1A1LMNASLC6A2SLC6A3RAB9A
SCHEMBL8154820 0.70 ALDH1A1 (0.39) ALDH1A1LMNAGAASLC6A2SLC6A3
SCHEMBL28513170 0.68 HPGD (0.32) MAPTHPGDHTT
SCHEMBL15680018 0.66 CES2 (0.63) ALDH1A1LMNAHPGDCES2CES1
SCHEMBL5444935 0.66 CES2 (0.63) ALDH1A1LMNAHPGDCES2CES1
SCHEMBL12763852 0.66
SCHEMBL7508732 0.66 NPC1 (0.36) ALDH1A1LMNASLC6A2SLC6A3RAB9A
SCHEMBL2297437 0.65 ALDH1A1 (0.53) ALDH1A1LMNACES2CES1KDM4E
SCHEMBL5781172 0.65 MMP2 (0.38) ALDH1A1LMNASLC6A2SLC6A3MAPT
SCHEMBL7550562 0.65 ALOX5 (0.41) SLC6A2SLC6A3CES2CES1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed