SCHEMBL8549059

SCHEMBL8549059

CCOC(=O)c1c(C2CC2)nc(CC)n1Cc1c2ccocc-2c(Cl)c1-c1ccccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
TSHR P16473 2/20 0.38
SIRT3 Q9NTG7 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
ADORA2B P29275 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545688 0.91 ALDH1A1 (0.38) ALDH1A1TSHRSIRT3ADORA2BMAPT
SCHEMBL9665278 0.91
SCHEMBL8545039 0.90 ALDH1A1 (0.37) ALDH1A1TSHRADORA2BMAPTLMNA
SCHEMBL8550121 0.85 ALDH1A1 (0.34) ALDH1A1TSHRMEN1KMT2ABUB1
SCHEMBL8544134 0.85
SCHEMBL9429570 0.83 ALDH1A1 (0.38) ALDH1A1TSHRAGTR1AGTR2
SCHEMBL8544609 0.82 TSHR (0.38) ALDH1A1TSHRMAPTLMNAHTT
SCHEMBL9663223 0.81 AGTR1 (0.30) AGTR1AGTR2
SCHEMBL9310339 0.81 KDM4E (0.33) ALDH1A1SIRT3CYP1A2CYP2C9CYP2C19
SCHEMBL9663265 0.80 GRM2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514198-B1 1H-Imidazol-1-yl-methyl benzofuran derivatives with the imidazolyl moiety being substituted by a cycloalkyl group GLAXO GROUP LTD (GB) 1998-08-05 EP disclosed
US-5498722-A HYPOTENSIVES GLAXO GROUP (GB) 1996-03-12 US disclosed
US-5332831-A Angiotensin antagonist GLAXO GROUP LIMITED (GB) 1994-07-26 US disclosed
WO-1992020674-A1 1H-IMIDAZOL-1-YL-METHYL BENZOFURAN DERIVATIVES, WITH THE IMIDAZOLYL MOIETY BEING SUBSTITUTED BY A CYCLOALKYL GROUP GLAXO GROUP LIMITED (GB) 1992-11-26 WO disclosed