SCHEMBL8549128

SCHEMBL8549128

O=C(CN1CCC[C@@H]1C(=O)NC(=O)c1ccccc1)OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.48
MMEL1 Q495T6 1/20 0.48
CTRB1 P17538 1/20 0.45
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
HSD17B10 Q99714 1/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
ACE P12821 2/20 0.43
HDAC3 O15379 1/20 0.43
FKBP1A P62942 2/20 0.43
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACE2 Q9BYF1 1/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549125 1.00 NPSR1 (0.48) NPSR1MMEL1CTRB1MMP2MMP9
SCHEMBL8545024 0.86 ALDH1A1 (0.45) NPSR1ACEALDH1A1SMN1; SMN2MAPT
SCHEMBL8545028 0.86 ALDH1A1 (0.45) NPSR1ACEALDH1A1SMN1; SMN2MAPT
SCHEMBL8549131 0.84 FKBP1A (0.55) MMEL1HDAC1HDAC2HDAC3FKBP1A
SCHEMBL8544794 0.83 NPSR1 (0.47) NPSR1ACEALDH1A1MAPT
SCHEMBL14836855 0.83 MMEL1 (0.52) MMEL1CTRB1ACEFKBP1AALDH1A1
SCHEMBL8544789 0.83 NPSR1 (0.47) NPSR1ACEALDH1A1MAPT
SCHEMBL8543316 0.82 CTSK (0.53) NPSR1ALDH1A1KMT2AMAPT
SCHEMBL8543314 0.82 CTSK (0.53) NPSR1ALDH1A1KMT2AMAPT
SCHEMBL8546776 0.82 CTSK (0.42) NPSR1MMEL1ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
JP-6041064-A None JP disclosed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
JP-H0641064-A 2-OXOETHYL DERIVATIVE MILES INC 1994-02-15 JP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed