SCHEMBL8549240

SCHEMBL8549240

CC(C)c1oc2ccc(C(=O)N3CCN(c4ccccc4)CC3)cc2c1CCN(C)Cc1cccc2ncncc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
TSHR P16473 4/20 0.37
ALOX15 P16050 2/20 0.36
LMNA P02545 5/20 0.36
MAPT P10636 4/20 0.36
MAPK1 P28482 2/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 3/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 2/20 0.36
HPGD P15428 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
GFER P55789 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MGLL Q99685 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HTT P42858 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553478 0.85 MAPT (0.37) ALDH1A1TSHRALOX15LMNAMAPT
SCHEMBL8192418 0.85 HSP90AA1 (0.38) ALDH1A1TSHRALOX15LMNAMAPT
SCHEMBL8552755 0.77 KDM4E (0.43) ALDH1A1LMNAMAPTGAAMEN1
SCHEMBL8551076 0.70 CNR2 (0.41) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL8552959 0.69 KDM4E (0.43) ALDH1A1LMNAMAPTPOLBGAA
Hexanoate SCHEMBL8550591 0.63 CNR2 (0.39) ALDH1A1TSHRMAPTUSP2POLB
SCHEMBL8708853 0.61 CNR2 (0.41) ALDH1A1MAPTPOLBHPGDGFER
SCHEMBL8197371 0.61 NPC1 (0.49) ALDH1A1HPGDGFERMEN1KMT2A
SCHEMBL8552304 0.60 CA9 (0.39)
SCHEMBL7141353 0.59 HTR1F (0.36) ALDH1A1LMNAMAPTMAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed