SCHEMBL8549348

SCHEMBL8549348

O=C1CCc2cccc(C(O)CCN3CCC(Cc4ccccc4)CC3)c2N1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.53
ADRA1D P25100 2/20 0.53
ADRA1A P35348 2/20 0.53
ADRA1B P35368 2/20 0.53
GRIN2D O15399 1/20 0.53
GRIN3B O60391 1/20 0.53
GRIN1 Q05586 1/20 0.53
GRIN2A Q12879 1/20 0.53
GRIN2C Q14957 1/20 0.53
GRIN3A Q8TCU5 1/20 0.53
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
ADRB2 P07550 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
ADRB1 P08588 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD2 P14416 1/20 0.47
CHRM3 P20309 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547677 0.90 CARM1 (0.47) GRIN2BADRA1DADRA1AADRA1BGRIN2D
SCHEMBL8547315 0.84 GRIN2B (0.51) GRIN2BADRA1DADRA1AADRA1BGRIN2D
SCHEMBL8540534 0.83 CARM1 (0.43) GRIN2BMAOAMAOBMEN1KMT2A
SCHEMBL8547312 0.81 MAOA (0.54) GRIN2BADRA1DADRA1AADRA1BGRIN2D
SCHEMBL7305064 0.80 CHRM2 (0.46) GRIN2BMAOAMAOBCHRM2CHRM4
SCHEMBL8549343 0.80 GRIN2B (0.59) GRIN2BADRA1DADRA1AADRA1BGRIN2D
SCHEMBL8542975 0.79 MAOA (0.49) GRIN2BADRA1DADRA1AADRA1BMAOA
SCHEMBL11071104 0.77 MAOA (0.61) ADRA1DADRA1AADRA1BMAOAMAOB
SCHEMBL11069444 0.76 DRD4 (0.62) ADRB2ADRB1DRD2DRD4MEN1
SCHEMBL8543860 0.76 LMNA (0.37) GRIN2BMEN1KMT2ACCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed