SCHEMBL8549896

SCHEMBL8549896

CN(C)CCOc1cc([N+](=O)[O-])cc2c1OCC2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
CYP19A1 P11511 6/20 0.38
KCNH2 Q12809 3/20 0.36
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
REN P00797 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750822 0.80 CHRNB2 (0.44) CHRNB2CHRNA4ESR1ESR2KDM4E
SCHEMBL8550551 0.78 HTR1B (0.41) ESR1ESR2KDM4EHTR1DHTR1B
SCHEMBL21588916 0.76 CYP19A1 (0.48) CYP19A1MEN1KMT2A
SCHEMBL29814530 0.76 CYP19A1 (0.48) CYP19A1MEN1KMT2A
SCHEMBL8551515 0.76 ALDH1A1 (0.43) CHRNB2CHRNA4ESR1ESR2MEN1
SCHEMBL29814593 0.74 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL21588776 0.74 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL4753173 0.74 MAPT (0.41) CHRNB2CHRNA4KDM4EGAACYP19A1
SCHEMBL8549856 0.73 ALDH1A1 (0.33) CHRNB2CHRNA4ESR1ESR2MEN1
SCHEMBL7484667 0.71 ALDH1A1 (0.42) HTR1DHTR1BCYP19A1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736025-B1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-07-22 EP disclosed
US-5700818-A Dihydrobenzofuranyl-biphenyl carboxamides having 5HT1D antagonistic activity SMITHKLINE BEECHAM P.L.C. (GB) 1997-12-23 US disclosed