SCHEMBL8551515

SCHEMBL8551515

CN(C)CCNc1cc([N+](=O)[O-])cc2c1OCC2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
NPSR1 Q6W5P4 1/20 0.43
BCHE P06276 2/20 0.37
ACHE P22303 2/20 0.37
HTT P42858 2/20 0.36
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
KAT2B Q92831 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549896 0.76 CHRNB2 (0.45) ALDH1A1MEN1KMT2AESR1ESR2
SCHEMBL8549856 0.73 ALDH1A1 (0.33) ALDH1A1HTTPOLBSMN1; SMN2MEN1
SCHEMBL7484667 0.71 ALDH1A1 (0.42) ALDH1A1ACHEHTTSMN1; SMN2MEN1
SCHEMBL10580640 0.70 ALDH1A1 (0.41) ALDH1A1HTTPOLBSMN1; SMN2MEN1
SCHEMBL1064809 0.69 ALDH1A1 (0.47) ALDH1A1NPSR1BCHEACHEHTT
SCHEMBL1979879 0.68 PARP1 (0.41) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL29814297 0.68 GPR35 (0.43) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL8550301 0.68 GPR35 (0.41) ALDH1A1HTTPOLBSMN1; SMN2MEN1
SCHEMBL15427979 0.68 ALDH1A1 (0.48) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL8550097 0.68 GPR35 (0.43) ALDH1A1HTTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736025-B1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-07-22 EP disclosed
US-5700818-A Dihydrobenzofuranyl-biphenyl carboxamides having 5HT1D antagonistic activity SMITHKLINE BEECHAM P.L.C. (GB) 1997-12-23 US disclosed
EP-0736025-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT 1D? ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1996-10-09 EP disclosed
WO-1995017401-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-06-29 WO disclosed