SCHEMBL8550223

SCHEMBL8550223

NC(=O)N(O)Cc1ccc(Cc2ccc(CN(O)C(N)=O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 10/20 0.56
PLA2G10 O15496 1/20 0.44
PLA2G2A P14555 1/20 0.44
KMT2A Q03164 1/20 0.40
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
RIPK1 Q13546 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9372536 0.83 ALOX5 (0.53) ALOX5KMT2A
SCHEMBL6037547 0.83 ALOX5 (0.56) ALOX5RIPK1
SCHEMBL8546442 0.82 ALOX5 (0.51) ALOX5KMT2A
SCHEMBL7217220 0.77 LOXL2 (0.52) ALOX5KMT2A
SCHEMBL8550197 0.77 MMP2 (0.49) ALOX5KMT2A
SCHEMBL8549962 0.76 ITGB3 (0.49) ALOX5
SCHEMBL8545311 0.76 ITGB3 (0.49) ALOX5
SCHEMBL8546769 0.76 ITGB3 (0.49) ALOX5
SCHEMBL9162595 0.76 POLB (0.53) ALOX5KMT2A
SCHEMBL8547601 0.75 ALOX5 (0.46) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed